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检索条件"主题词=SynthesisAntifungalWater-soluble prodrugsltraconazole analogue"
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Synthesis,pharmacokinetics and in vivo antifungal activity of the novel water-soluble prodrugs of itraconazole analogue YL-24
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Chinese Chemical Letters 2013年 第4期24卷 321-324页
作者: Yu Liu Xu-Feng Cao Xin Liu Yong-Bing Cao Wen-Jing Chu Yu-She Yang State Key Laboratory of Drug Research Shanghai Institute of Materia MedicaChinese Academy of Sciences School of Pharmacy Second Military Medical University State Key Laboratory of Drug Research Shanghai Institute of Materia MedicoChinese Academy of Sciences
To improve the aqueous solubility of an itraconazole analogue, compound 1 (YL-24), a series of novel prodrugs were synthesized. Among these prodrugs, the phosphate disodium salt compound 7 exhibited excellent aqueou... 详细信息
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