Selective mono-arylation in palladium-catalyzed cross-coupling reaction of dichlorotriazines with phenylboronate ester derivatives
Selective mono-arylation in palladium-catalyzed cross-coupling reaction of dichlorotriazines with phenylboronate ester derivatives作者机构:School of Pharmaceutical SciencesCentral South University School of Pharmaceutical SciencesSun Yat-sen University
出 版 物:《Chinese Chemical Letters》 (中国化学快报(英文版))
年 卷 期:2013年第24卷第1期
页 面:41-44页
核心收录:
学科分类:081705[工学-工业催化] 08[工学] 0817[工学-化学工程与技术] 0703[理学-化学]
基 金:the National Natural Science Foundation of China(Nos.30873137 30772645 and 81172927) for their financial support
主 题:Suzuki cross coupling reactionDichlorotriazinesAryl boronic estersPd(PPh3)4
摘 要:Palladium-catalyzed cross-coupling reaction between dichlorotriazines and phenylboronate esters produced the mono-awlated triazines selectively and thus, the corresponding phenyltriazine derivatives could be assembled efficiently in moderate to good overall yields (50-80%).